发明名称 SALT OF 1-(2-DEOXY-2-FLUORO-4-THIO-beta-D-ARABINOFURANOSYL)CYTOSINE
摘要 A superior antitumor agent is provided. A salt of 1-(2-deoxy-2-fluoro-4-thio-²-D-arabinofuranosyl)cytosine shows at least one or more of such characteristics as (1) it has superior antitumor activity, (2) it shows superior crystallinity, (3) it shows high water solubility, (4) it does not show deliquescent property, (5) it shows superior flowability, (6) it shows superior tableting property, (7) it can be manufactured with less environmental load, and (8) it can be manufactured in a large scale, and therefore it is useful as a bulk drug for medicaments.
申请公布号 EP2832740(A4) 申请公布日期 2015.11.11
申请号 EP20130770090 申请日期 2013.03.27
申请人 FUJIFILM CORPORATION 发明人 BABA, YASUTAKA;MURAKAMI, TATSUYA;SHINTANI, JUNKO
分类号 C07H19/06;A61K31/7068;A61P35/00;C07C309/04;C07H19/073 主分类号 C07H19/06
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