| 发明名称 |
PROCESS FOR THE PREPARATION OF (2R,3S)-3-PHENYLISOSERINE METHYL ESTER ACETATE SALT |
| 摘要 |
<p>A process for the enantioselective preparation of (2R,3S)-3-phenylisoserine methyl ester acetate salt of formula (I) which is an useful building block for the synthesis of taxane derivatives. The process involves the resolution of racemic threo-phenylisoserine amide and its conversion into (I).</p> |
| 申请公布号 |
CA2679159(C) |
申请公布日期 |
2015.11.03 |
| 申请号 |
CA20082679159 |
申请日期 |
2008.02.11 |
| 申请人 |
INDENA S.P.A. |
发明人 |
CICERI, DANIELE;GABETTA, BRUNO;VIGNOLA, NICOLA;MITZEL, FRIEDER;WEBER, BEAT T. |
| 分类号 |
C07C237/20;C07C227/18;C07C227/30;C07C229/34 |
主分类号 |
C07C237/20 |
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