FUSED TRICYCLIC DUAL INHIBITORS OF CDK 4/6 AND FLT3
摘要
Compounds of Formula IIIA are useful inhibitors of CDK 4, CDK6, and FLT3. Such compounds are useful in treating cancer and various other disease conditions.
申请公布号
EP2937349(A1)
申请公布日期
2015.10.28
申请号
EP20150161337
申请日期
2012.03.21
申请人
AMGEN INC.
发明人
CHEN, XIAOQI;DAI, KANG;DUQUETTE, JASON A.;GRIBBLE, MICHAEL W., JR.;HUARD, JUSTIN N.;KEEGAN, KATHLEEN S.;LI, ZHIHONG;LIVELY, SARAH E.;MCGEE, LAWRENCE R.;RAGAINS, MARK L.;WANG, XIANGHONG;WEIDNER, MARGARET F.;ZHANG, JIAN