COMPOUND; TAUTOMER AND GEOMETRIC ISOMER THEREOF; SALT OF SAID COMPOUND, TAUTOMER, OR GEOMETRIC ISOMER; METHOD FOR MANUFACTURING SAID COMPOUND, TAUTOMER, ISOMER, OR SALT; ANTIMICROBIAL AGENT; AND ANTI-INFECTIVE DRUG

摘要

The present invention provides compounds belonging to 3-acyloxyindole compounds or 3-acyl-4-hydroxycoumarin compounds, a tautomer or geometric isomer thereof, or a salt thereof and methods for producing the same, which compounds are useful as antibacterial agent and as therapeutic drugs against infectious diseases.

主权项

1. A compound represented by any one of General Formulas (1) to (2) below, a tautomer or geometric isomer thereof, or a salt thereof: wherein X1 represents a single bond or an alkylene group having 1 to 8 carbon atoms, Y1 represents a single bond, —O—, —NHCO—, —NHCOO—, —S—, —SO—, or —SO2—, Z1 represents a cyclic, linear, or branched alkyl group which has 8 to 30 carbon atoms and may have a halogen atom, X2 represents a single bond, —CO—, —CONH—, or —COO—, Y2 represents a hydrocarbon group which has 1 to 30 carbon atoms and may have —CN, —NO2, an alkoxy group, a halogen atom, or any combination thereof; or a hydrogen atom, X3 represents a single bond or —NH—, Z represents a hydrogen atom, a halogen atom, an alkoxy group having 1 to 6 carbon atoms, or a hydrocarbon group having 1 to 20 carbon atoms, and R1 represents a hydrocarbon group which has 1 to 30 carbon atoms and may have an alkoxy group, —OH, —CN, —NO2, a halogen atom, or any combination thereof.