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发明名称
Process for the preparation of nebivolol
摘要
<p>The present invention relates to a novel process for the synthesis of the Nebivolol product depicted in Scheme 1, comprised of a reduced number of high-yield steps, and characterized by the enzymatic resolution of the chroman ester precursor.</p>
申请公布号
EP2646426(B1)
申请公布日期
2015.10.07
申请号
EP20110815574
申请日期
2011.11.30
申请人
MENARINI INTERNATIONAL OPERATIONS LUXEMBOURG S.A.
发明人
MAURO, SANDRO;FATTORI, DANIELA;D'ANDREA, PIERO;CIPOLLONE, AMALIA
分类号
C07D311/58;C12P17/16
主分类号
C07D311/58
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代理人
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