发明名称 BILE ACID DERIVATIVES AS FXR LIGANDS FOR THE PREVENTION OR TREATMENT OF FXR-MEDIATED DESEASES OR CONDITIONS
摘要 The present invention relates to compounds of formula (I) wherein R is hydrogen or alpha-hydroxy, the hydroxyl group in position 7 is in the alpha or beta position; and pharmaceutically acceptable salts, solvates or amino acid conjugates thereof.
申请公布号 WO2008002573(A3) 申请公布日期 2008.02.28
申请号 WO2007US14829 申请日期 2007.06.27
申请人 INTERCEPT PHARMACEUTICALS, INC.;PELLICCIARI, ROBERTO;FIORUCCI, STEFANO;PRUZANSKI, MARK 发明人 PELLICCIARI, ROBERTO;FIORUCCI, STEFANO;PRUZANSKI, MARK
分类号 C07J9/00;A61K31/575 主分类号 C07J9/00
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