发明名称 | Heteroaryl carboxamides | ||
摘要 | The invention relates to novel heteroaryl carboxamides, a process for their preparation, and pharmaceutical compositions containing them. These materials are useful for the treatment and/or prophylaxis of diseases and for improving perception, concentration, learning and/or memory. | ||
申请公布号 | US9139579(B2) | 申请公布日期 | 2015.09.22 |
申请号 | US201213544321 | 申请日期 | 2012.07.09 |
申请人 | BAYER INTELLECTUAL PROPERTY GMBH | 发明人 | Hendrix Martin;Böβ Frank-Gerhard;Erb Christina;Krüger Joachim;Luithle Joachim;Methfessel Christoph;Schreiber Rudy;Wiese Welf-Burkhard |
分类号 | C07D453/02 | 主分类号 | C07D453/02 |
代理机构 | Locke Lord LLP | 代理人 | Locke Lord LLP ;DiCeglie, Jr. Nicholas J. |
主权项 | 1. A compound of the formula (I): in which R1 is 1-azabicyclo[2.2.2]oct-3-yl, the ring A is pyridazino, and R2 and R3 are identical or different and are radicals selected from the group of hydrogen, halogen, formyl, carbamoyl, cyano, trifluoromethyl, trifluoromethoxy, nitro, (C1-C6)-alkyl , (C1-C6)-alkoxy, (C1-C6)-alkylthio, (C3-C8)-cycloalkyl, 4- to 8-membered heterocyclyl, phenyl or 5- to 6-membered heteroaryl, where phenyl and heteroaryl are optionally substituted by halogen, (C1-C4)-alkyl, (C1-C4)-alkoxy, amino, mono- or di-(C1-C4)-alkylamino, (C1-C4)-alkanoylamino or (C1-C4) -alkanesulfonylamino; or a salt thereof. | ||
地址 | Monheim DE |