Tubulysins are a series of naturally occurring cytotoxic agents that are of interest as anticancer therapeutic agents. Processes and intermediates useful for preparing naturally occurring and non-naturally occurring tubulysins and analogs and derivatives thereof are described.
申请公布号
AU2011285532(B2)
申请公布日期
2015.09.10
申请号
AU20110285532
申请日期
2011.08.05
申请人
ENDOCYTE, INC.
发明人
VLAHOV, IONTCHO RADOSLAVOV;GROANING, MICHAEL;KLEINDL, PAUL JOSEPH;SANTHAPURAM, HARI KRISHNA R.;YOU, FEI;WANG, YU;XU, LE-CUN;STANFORD, KATHERYN MARIE;RITTER, ALLEN;LEAMON, CHRISTOPHER PAUL