发明名称 4-SUBSTITUENT-2-HYDROXYLMORPHOLINE-3-ONE AND PREPARATION METHOD THEREOF
摘要 <p>A molecule with neural activities, especially 4-substituent-2-hydroxymorpholin-3-one, as a new intermediate of neurokinin-1 receptor antagonist aprepitant, and preparation method thereof.</p>
申请公布号 EP2837624(A4) 申请公布日期 2015.09.09
申请号 EP20130775919 申请日期 2013.04.15
申请人 ZHEJIANG HISUN PHARMACEUTICAL CO. LTD.;SHANGHAI INSTITUTE OF PHARMACEUTICAL INDUSTRY 发明人 ZHANG, FULI;LIU, CHONGHAO;QIU, PENGCHENG;CHAI, JIAN;CAI, QINGFENG
分类号 C07D265/32;C07D413/06 主分类号 C07D265/32
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