| 主权项 |
1. A 3-phenylisoxazoline derivative and/or salt thereof, of formula (I) in which R1 and R2 are each independently hydrogen, fluorine, chlorine, bromine, iodine, cyano, or (C1-C4)-alkyl or (C1-C4)-alkoxy each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine and cyano, or R1 and R2 together with the carbon atom to which they are bonded form a saturated or partly or fully unsaturated three-, four- or five-membered ring formed from q carbon atoms and p oxygen atoms; R3 is fluorine, chlorine, cyano, (C1-C3)-alkylcarbonyloxy or S(O)nR5, or (C1-C6)-alkyl, (C3-C6)-cycloalkyl, (C2-C6)-alkenyl or (C2-C6)-alkynyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano, (C1-C4)-alkoxy and hydroxyl, or (C1-C6)-alkylcarbonyl, (C2-C6)-alkenylcarbonyl or (C3-C6)-cycloalkylcarbonyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and (C1-C6)-alkoxy; R5 is (C1-C6)-alkyl or (C3-C6)-cycloalkyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and hydroxyl; R6 is hydrogen or R5; R7 is hydrogen or (C1-C6)-alkyl, (C3-C6)-cycloalkyl, (C2-C4)-alkenyl or (C2-C4)-alkynyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, cyano and (C1-C2)-alkoxy; R8 is R7; W* is COOH, COOY, CN or CHO; Y is (C1-C8)-alkyl which is substituted by m radicals from the group consisting of fluorine, chlorine, bromine, cyano, hydroxyl and COO—(C1-C8)-alkyl and which is interrupted by n heteroatoms from the group consisting of oxygen, sulfur and nitrogen, or a radical from the group consisting of (cyclohex-2-en-1-one)-3-yl, (propan-1-ol)-3-yl, (2,2-dimethylpropan-1-ol)-3-yl, (methyl 2,2-dimethylpropanoate)-3-yl, (methyl propanoate)-3-yl, (ethyl propanoate)-3-yl, (ethyl butanoate)-3-yl, (ethyl (3R)-4,4,4-trifluorobutanoate)-3-yl, (butan-2-one)-4-yl, (3-methylbutan-2-one)-4-yl, (pent-3-en-2-one)-4-yl, ((2S)-dimethyl butanedioate)-2-yl, (dimethyl pentanedioate)-3-yl, (methyl (2R)-2-methylpropanoate)-3-yl, 4-methoxycarbonylbenzyl, 3,5-difluorobenzyl, 3,4-difluorobenzyl, 2,6-difluorobenzyl, 5-methylpyridin-3-ylmethyl, tetrahydrofuran-3-yl and (butan-1-ol)-4-yl; X2, X4 and X6 are each independently hydrogen, fluorine, chlorine, bromine, iodine, cyano, nitro, or (C1-C4)-alkyl, (C3-C5)-cycloalkyl, (C2-C4)-alkenyl, (C2-C4)-alkynyl, (C1-C4)-alkoxy, (C2-C4)-alkenyloxy, (C2-C4)-alkynyloxy or (C1-C4)-alkylcarbonyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and (C1-C4)-alkoxy; X3 is fluorine, chlorine, bromine, iodine, hydroxyl, cyano, nitro, SF5, CONR8SO2R5, CONR6R8, CORE, CO2R8, CONR6R8, C(R6)═NOR8, NR6COR8, NR6CONR8R8, NR6CO2R8, NR6SO2R8, NR6SO2NR6R8, OCONR6R8, OSO2R5, R5, S(O)nR5, SO2NR6R8, OSO2NR6R8, or (C1-C6)-alkyl, (C3-C5)-cycloalkyl, (C2-C6)-alkenyl, (C2-C6)-alkynyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, hydroxyl and cyano, or (C1-C6)-alkoxy, (C3-C6)-cycloalkoxy, (C2-C6)-alkenyloxy or (C2-C6)-alkynyloxy each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and (C1-C2)-alkoxy; X5 is hydrogen, fluorine, chlorine, bromine, iodine, hydroxyl, cyano, nitro, SF5, CONR8SO2R5, CONR6R8, CORE, CO2R8, CONR6R8, C(R6)═NOR8, NR6COR8, NR6CONR8R8, NR6CO2R8, NR6SO2R8, NR6SO2NR6R8, OCONR6R8, OSO2R5, R5, S(O)nR5, SO2NR6R8, OSO2NR6R8, or (C1-C6)-alkyl, (C3-C5)-cycloalkyl, (C2-C6)-alkenyl, (C2-C6)-alkynyl each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, hydroxyl and cyano, or (C1-C6)-alkoxy, (C3-C6)-cycloalkoxy, (C2-C6)-alkenyloxy or (C2-C6)-alkynyloxy each substituted by m radicals from the group consisting of fluorine, chlorine, bromine, iodine, cyano and (C1-C2)-alkoxy; m is 0, 1, 2, 3, 4 or 5; n is 0, 1 or 2; p is 0 or 1; q is 3, 4 or 5; with the proviso that a) X3 and X4 are not both substituted or unsubstituted alkoxy, b) in the compounds in which R3 is methyl and W* is COOH, X5 is not hydrogen, and c) the compounds methyl 3-(3-cyanophenyl)-5-(isopropoxymethyl)-4,5-dihydro-1,2-oxazole-5-carboxylate, methyl 5-(butoxymethyl)-3-(3-cyanophenyl)-4,5-dihydro-1,2-oxazole-5-carboxylate, methyl 3-(3-cyanophenyl)-5-(methoxymethyl)-4,5-dihydro-1,2-oxazole-5-carboxylate, methyl 3-(3-cyanophenyl)-5-(2-methoxyethyl)-4,5-dihydro-1,2-oxazole-5-carboxylate, 3-(3-cyanophenyl)-5-(trifluoromethyl)-4,5-dihydro-1,2-oxazole-5-carboxylic acid, methyl 3-(3-cyanophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate, ethyl 3-(3-cyanophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate, methyl 5-methyl-3-(3-nitrophenyl)-4,5-dihydro-1,2-oxazole-5-carboxylate, methyl 3-(3,5-di-tert-butyl-4-hydroxyphenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate and ethyl 3-(3-chlorophenyl)-5-methyl-4,5-dihydro-1,2-oxazole-5-carboxylate are excluded. |
