发明名称 |
POLYMER COMPOUND HAVING CAMPTOTHECIN DERIVATIVE AND HSP90 INHIBITOR BONDED THERETO, AND USE THEREFOR |
摘要 |
Provided are: a polymer compound for efficiently delivering two drugs to an affected area, reducing side effects, and increasing drug efficacy; and an antitumor drug having said polymer compound as an active ingredient. This polymer compound is obtained by ester-bonding a camptothecin derivative and an HSP90 inhibitor to a carboxyl group of a side-chain of a block copolymer obtained by joining a polyethylene glycol segment and a polyglutamic acid segment to one another. |
申请公布号 |
WO2015125640(A1) |
申请公布日期 |
2015.08.27 |
申请号 |
WO2015JP53479 |
申请日期 |
2015.02.09 |
申请人 |
NIPPON KAYAKU KABUSHIKI KAISHA |
发明人 |
OKAZAKI MANAMI;MARUYAMA SAKIKO;MASUDA AKIRA;YAMAMOTO KEIICHIRO |
分类号 |
A61K47/48;A61K31/4196;A61K31/4745;A61K45/00;A61K47/34;A61P35/00;A61P43/00;C08G69/40 |
主分类号 |
A61K47/48 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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