发明名称 POLYMER COMPOUND HAVING CAMPTOTHECIN DERIVATIVE AND HSP90 INHIBITOR BONDED THERETO, AND USE THEREFOR
摘要 Provided are: a polymer compound for efficiently delivering two drugs to an affected area, reducing side effects, and increasing drug efficacy; and an antitumor drug having said polymer compound as an active ingredient. This polymer compound is obtained by ester-bonding a camptothecin derivative and an HSP90 inhibitor to a carboxyl group of a side-chain of a block copolymer obtained by joining a polyethylene glycol segment and a polyglutamic acid segment to one another.
申请公布号 WO2015125640(A1) 申请公布日期 2015.08.27
申请号 WO2015JP53479 申请日期 2015.02.09
申请人 NIPPON KAYAKU KABUSHIKI KAISHA 发明人 OKAZAKI MANAMI;MARUYAMA SAKIKO;MASUDA AKIRA;YAMAMOTO KEIICHIRO
分类号 A61K47/48;A61K31/4196;A61K31/4745;A61K45/00;A61K47/34;A61P35/00;A61P43/00;C08G69/40 主分类号 A61K47/48
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