发明名称 A NEW METHOD FOR PRODUCING NEBIVOLOL HYDROCHLORIDE OF HIGH PURITY
摘要 The invention relates to a process for producing Nebivolol hydrochloride, (formula I) comprising the steps of: provision of a protected Nebivolol hydrochloride of the general formula (II), with P being an amine protecting group, and hydrogenation of said protected Nebivolol hydrochloride yielding Nebivolol hydrochloride of the formula (I).
申请公布号 CA2937826(A1) 申请公布日期 2015.08.20
申请号 CA20152937826 申请日期 2015.02.13
申请人 CORDEN PHARMA INTERNATIONAL GMBH 发明人 CLAVEL, ALEXANDRE;FREIFELD, DR. ILIA;JAS, DR. GERHARD;KESSELER, DR. KURT
分类号 C07D311/58 主分类号 C07D311/58
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