发明名称 GUANIDINE AND AMINE SUBSTITUTED TETRAHYDROISOQUINOLINE COMPOUNDS AS FACTOR XIA INHIBITORS
摘要 The present invention provides compounds of Formula (I): (Formula (I)) or stereoisomers, pharmaceutically acceptable salts thereof, wherein all of the variables are as defined herein. These compounds are inhibitors of factor XIa and/or plasma kallikrein which may be used as medicaments.
申请公布号 EP2906541(A1) 申请公布日期 2015.08.19
申请号 EP20130780043 申请日期 2013.10.11
申请人 BRISTOL-MYERS SQUIBB COMPANY 发明人 PINTO, DONALD J. P.;CLARK, CHARLES G.;ORWAT, MICHAEL J.;SMITH II, LEON M.;EWING, WILLIAM R.
分类号 C07D217/26;A61K31/472;A61K31/4725;A61P7/02;C07D401/04;C07D405/04;C07D409/04 主分类号 C07D217/26
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