发明名称 |
GUANIDINE AND AMINE SUBSTITUTED TETRAHYDROISOQUINOLINE COMPOUNDS AS FACTOR XIA INHIBITORS |
摘要 |
The present invention provides compounds of Formula (I): (Formula (I)) or stereoisomers, pharmaceutically acceptable salts thereof, wherein all of the variables are as defined herein. These compounds are inhibitors of factor XIa and/or plasma kallikrein which may be used as medicaments. |
申请公布号 |
EP2906541(A1) |
申请公布日期 |
2015.08.19 |
申请号 |
EP20130780043 |
申请日期 |
2013.10.11 |
申请人 |
BRISTOL-MYERS SQUIBB COMPANY |
发明人 |
PINTO, DONALD J. P.;CLARK, CHARLES G.;ORWAT, MICHAEL J.;SMITH II, LEON M.;EWING, WILLIAM R. |
分类号 |
C07D217/26;A61K31/472;A61K31/4725;A61P7/02;C07D401/04;C07D405/04;C07D409/04 |
主分类号 |
C07D217/26 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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