发明名称 |
IMIDAZOLINE DERIVATIVES, PREPARATION METHODS THEREOF, AND THEIR APPLICATIONS IN MEDICINE |
摘要 |
<p>New imidazoline derivatives represented by formula (I), preparation methods thereof, pharmaceutical compositions comprising such derivatives, and applications of such derivatives in preparing androgen receptor antagonists and medicaments for treating diseases such as prostate cancer.</p> |
申请公布号 |
EP2894151(A1) |
申请公布日期 |
2015.07.15 |
申请号 |
EP20130835193 |
申请日期 |
2013.08.26 |
申请人 |
SHANGHAI HENGRUI PHARMACEUTICAL CO. LTD.;JIANGSU HENGRUI MEDICINE CO. LTD. |
发明人 |
LU, HEJUN;SUN, PIAOYANG;FEI, HONGBO;JIANG, HONGJIAN;WANG, HAOWEI;DONG, QING |
分类号 |
C07D233/72;A61K31/4164;A61K31/4166;A61K31/4178;A61P5/28;A61P35/00;C07D233/84;C07D233/86 |
主分类号 |
C07D233/72 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|