发明名称 Process for the preparation of sulfonamide compounds
摘要 Process for the preparation of known sulfonamides having antibacterial activity applicable on industrial scale, which allows their production in high yields and purity, comprising in particular the step of nucleophile aromatic substitution and oxidation in suitable conditions.
申请公布号 US9079831(B2) 申请公布日期 2015.07.14
申请号 US201414243058 申请日期 2014.04.02
申请人 Dipharma Francis S.r.l. 发明人 Allegrini Pietro;Mantegazza Simone
分类号 C07C213/00;C07C315/02;C07C317/14;C07C317/36;C07C323/09;C07C319/18 主分类号 C07C213/00
代理机构 Rothwell, Figg, Ernst & Manbeck, P.C. 代理人 Rothwell, Figg, Ernst & Manbeck, P.C.
主权项 1. A process for preparing a compound of formula (I) comprising reacting a compound of formula (II) with a compound of formula (III) wherein R is a C1-C6 alkyl group or phenyl group, in the presence of a base and in a solvent.
地址 Baranzate (MI) IT