发明名称 |
PROCESS FOR PREPARATION OF ABIRATERONE ACETATE |
摘要 |
The present invention relates to improvement in the process of preparation of abiraterone acetate or a pharmaceutically acceptable salt thereof wherein the improvement comprises purifying the crude 3-?-acetoxyandrosta-5,16-diene-17-yl trifluoromethane sulphonate by crystallization from a solvent to obtain acetoxyandrosta-5,16-diene-17-yl trifluoromethane sulphonate as a crystalline solid and converting it to abiraterone acetate or pharmaceutically acceptable salt thereof. |
申请公布号 |
IN2133MU2013(A) |
申请公布日期 |
2015.06.05 |
申请号 |
IN2013MUM2133 |
申请日期 |
2013.06.24 |
申请人 |
SUN PHARMACEUTICAL INDUSTRIES LTD. |
发明人 |
THENNATI RAJAMANNAR;REHANI RAJEEV BUDHDEV;PATEL NISCHALKUMAR VINODBHAI;KANSARA RITESHKUMAR RAJNIKANT |
分类号 |
C07J43/00;C07J13/00;C07J41/00 |
主分类号 |
C07J43/00 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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