发明名称 |
PROCESS AND INTERMEDIATES FOR THE PREPARATION OF ABIRATERONE ACETATE |
摘要 |
The present invention relates to a process for the synthesis of (3beta)17-(3-pyridinyl)androsta-5,16-dien-3-yl acetate (Abiraterone acetate) represented by the structure of formula (1), and salts thereof, especially salts with pharmaceutically acceptable acids. The present invention further relates to certain intermediates in such processes. |
申请公布号 |
EP2877482(A1) |
申请公布日期 |
2015.06.03 |
申请号 |
EP20130822913 |
申请日期 |
2013.07.22 |
申请人 |
MAPI PHARMA LIMITED |
发明人 |
MAROM, EHUD;RUBNOV, SHAI;MIZHIRITSKII, MICHAEL |
分类号 |
C07J43/00;A61K31/56;A61K31/58;A61P35/00;C07J51/00 |
主分类号 |
C07J43/00 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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