发明名称 |
Crystalline molecular comlpexes of tadalafil |
摘要 |
Crystalline molecular complexes of tadalafil are disclosed. The crystalline molecular complexes include those of tadalafil and oxalic acid, tadalafil and 4-hydroxybenzoic acid, tadalafil and 3-phenylpropanoic acid, tadalafil and malonic acid, tadalafil and methylparaben, and tadalafil and propylparaben. Pharmaceutical compositions containing the crystalline molecular complexes are also disclosed. |
申请公布号 |
US9040535(B2) |
申请公布日期 |
2015.05.26 |
申请号 |
US201314047463 |
申请日期 |
2013.10.07 |
申请人 |
THAR PHARMACEUTICALS, INC. |
发明人 |
Hanna Mazen;Shan Ning;Cheney Miranda L.;Weyna David R. |
分类号 |
A61K31/4985;C07D487/22;C07D471/14 |
主分类号 |
A61K31/4985 |
代理机构 |
J. A. Lindeman & Co., PLLC |
代理人 |
J. A. Lindeman & Co., PLLC |
主权项 |
1. A crystalline molecular complex of tadalafil comprising tadalafil and a propylparaben co-former. |
地址 |
Pittsburgh PA US |