发明名称 Crystalline molecular comlpexes of tadalafil
摘要 Crystalline molecular complexes of tadalafil are disclosed. The crystalline molecular complexes include those of tadalafil and oxalic acid, tadalafil and 4-hydroxybenzoic acid, tadalafil and 3-phenylpropanoic acid, tadalafil and malonic acid, tadalafil and methylparaben, and tadalafil and propylparaben. Pharmaceutical compositions containing the crystalline molecular complexes are also disclosed.
申请公布号 US9040535(B2) 申请公布日期 2015.05.26
申请号 US201314047463 申请日期 2013.10.07
申请人 THAR PHARMACEUTICALS, INC. 发明人 Hanna Mazen;Shan Ning;Cheney Miranda L.;Weyna David R.
分类号 A61K31/4985;C07D487/22;C07D471/14 主分类号 A61K31/4985
代理机构 J. A. Lindeman & Co., PLLC 代理人 J. A. Lindeman & Co., PLLC
主权项 1. A crystalline molecular complex of tadalafil comprising tadalafil and a propylparaben co-former.
地址 Pittsburgh PA US
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