发明名称 CRYSTALLINE FORM OF PRULIFLOXACIN AND PROCESSES FOR ITS PREPARATION
摘要 The present invention relates to a crystalline polymorphic form of 6-fluoro-1-methyl-7- {4-[(5-methyl-2-oxo-1,3-dioxol-4-yl)methyl]piperazin-1-yl}-4-oxo-4H-[1,3]-thiazeto-[3,2- a]-quinoline-3-carboxylic acid (prulifloxacin). More specifically, the invention relates to a crystalline form of prulifloxacin (herein referred to as Form A), and a method for preparing the crystalline Form A. The present invention further provides a pharmaceutical formulation comprising the novel form of prulifloxacin.
申请公布号 IN2925MUN2012(A) 申请公布日期 2015.05.22
申请号 IN2012MUMNP2925 申请日期 2012.12.31
申请人 CIPLA LIMITED 发明人 PATHI  SRINIVAS  LAXMINARAYAN;RAO&NBSP, DHARMARAJ&NBSP, RAMACHANDRA;KANKAN&NBSP, RAJENDRA;CHINIMILLI&NBSP, VENUGOPALARAO
分类号 C07D513/04;A61K31/496 主分类号 C07D513/04
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