| 摘要 |
The present invention relates to inhibitors of bromo and extra terminal (BET) bromodomains that are useful for the treatment of cancer, inflammatory diseases, diabetes, and obesity, having Formula (I): wherein W, X, Y, Z, R1, R2, R5, and R8 are as described herein. |
| 申请人 |
BAIR, KENNETH W.;HERBERTZ, TORSTEN;KAUFFMAN, GOSS STRYKER;KAYSER-BRICKER, KATHERINE J.;LUKE, GEORGE P.;MARTIN, MATTHEW W.;MILLAN, DAVID S.;SCHILLER, SHAWN E. R.;TALBOT, ADAM C. |
发明人 |
BAIR, KENNETH W.;HERBERTZ, TORSTEN;KAUFFMAN, GOSS STRYKER;KAYSER-BRICKER, KATHERINE J.;LUKE, GEORGE P.;MARTIN, MATTHEW W.;MILLAN, DAVID S.;SCHILLER, SHAWN E. R.;TALBOT, ADAM C. |
