| 主权项 |
1. An N-(1,2,5-oxadiazol-3-yl)-, N-(tetrazol-5-yl)- or N-(triazol-5-yl)bicycloarylcarboxamide of the formula (I) or a salt thereof in which Q is a Q1, Q2 or Q3 radical, R1 is (C1-C6)-alkyl, (C3-C7)-cycloalkyl, halo-(C1-C6)-alkyl, (C2-C6)-alkenyl, halo-(C2-C6)-alkenyl, (C2-C6)-alkynyl, halo-(C2-C6)-alkynyl, (C1-C6)-alkoxy-(C1-C6)-alkyl, (C1-C6)- alkoxy-(C2-C6)-alkenyl, (C1-C6)-alkoxy-(C2-C6)-alkynyl, CH2R6, heteroaryl, heterocyclyl or phenyl, where the three latter radicals are each substituted by u radicals from the group consisting of halogen, nitro, cyano, (C1-C6)-alkyl, halo-(C1-C6)-alkyl, (C3-C6)-cycloalkyl, (C1-C6)-alkylthio, (C1-C6)-alkylsulfinyl, (C1-C6)-alkylsulfonyl, (C1-C6)-alkoxy, halo-(C1-C6)-alkoxy and (C1-C6)-alkoxy-(C1-C4)-alkyl; R2 is hydrogen, (C1-C6)-alkyl, (C3-C7)-cycloalkyl, halo-(C1-C6)-alkyl, (C1-C6)-alkoxy, halo-(C1-C6)-alkoxy, (C2-C6)-alkenyl, (C2-C6)-alkenyloxy, halo-(C2-C6)-alkenyl, (C2-C6)-alkynyl, (C2-C6)-alkynyloxy, halo-(C2-C6)-alkynyl, cyano, nitro, methylsulfenyl, methylsulfinyl, methylsulfonyl, acetylamino, benzoylamino, methoxycarbonyl, ethoxycarbonyl, methoxycarbonylmethyl, ethoxycarbonylmethyl, benzoyl, methylcarbonyl, piperidinylcarbonyl, trifluoromethylcarbonyl, halogen, amino, aminocarbonyl, methylaminocarbonyl, dimethylaminocarbonyl, methoxymethyl, or heteroaryl, heterocyclyl or phenyl each substituted by u radicals selected from the group consisting of methyl, ethyl, methoxy, trifluoromethyl and halogen; R3 and R4 are each independently hydrogen, (C1-C6)-alkyl, halo-(C1-C6)-alkyl, (C2-C6)-alkenyl, halo-(C2-C6)-alkenyl, (C2-C6)-alkynyl, halo-(C2-C6)-alkynyl, (C3-C7)-cycloalkyl, (C3-C7)-halocycloalkyl, (C1-C6)-alkoxy, (C1-C6)-haloalkoxy, (C1-C6)-alkylthio, (C1-C6)-haloalkylthio, (C1-C6)-alkylsulfinyl, (C1-C6)-haloalkylsulfinyl, (C1-C6)-alkylsulfonyl, (C1-C6)-haloalkylsulfonyl, (C1-C6)-alkoxy-(C1-C4)-alkyl, halogen, nitro or cyano; R5 is hydrogen or fluorine; R6 is acetoxy, acetamido, N-methylacetamido, benzoyloxy, benzamido, N-methylbenz-amido, methoxycarbonyl, ethoxycarbonyl, benzoyl, methylcarbonyl, piperidinylcarbonyl, morpholinylcarbonyl, trifluoromethylcarbonyl, aminocarbonyl, methylaminocarbonyl, dimethylaminocarbonyl, (C3-C6)-cycloalkyl, or heteroaryl, heterocyclyl or phenyl each substituted by u radicals selected from the group consisting of methyl, ethyl, methoxy, trifluoromethyl and halogen; R7 and R8 are each independently hydrogen, (C1-C6)-alkyl, halo-(C1-C6)-alkyl, (C2-C6)-alkenyl, halo-(C2-C6)-alkenyl, (C2-C6)-alkynyl, halo-(C2-C6)-alkynyl, (C3-C7)-cycloalkyl, halo-(C3-C7) -cycloalkyl, -OR9, S(O)mR9, (C1-C6)-alkylthio, halo-(C1-C6)-alkylthio, (C1-C6)-alkylsulfinyl, halo-(C1-C6)-alkylsulfinyl, (C1-C6)-alkylsulfonyl, halo-(C1-C6)-alkyl-sulfonyl, (C1-C6)-alkoxy-(C1-C4)-alkyl, halogen, nitro, cyano, heteroaryl, heterocyclyl or phenyl, where the three latter radicals are each substituted by u radicals selected from the group consisting of halogen, nitro, cyano, (C1-C6)-alkyl, halo-(C1-C6)-alkyl, (C3-C6)-cycloalkyl, (C1-C6)-alkylthio, (C1-C6)-alkylsulfinyl, (C1-C6)-alkylsulfonyl, (C1-C6)- alkoxy, halo-(C1-C6)-alkoxy and (C1-C6)-alkoxy-(C1-C4)-alkyl, or R7 and R8 together with the carbon atom to which they are bonded form a —X1—(CH2)r—X2—, —(CH2)s—X3—, —(CH2)t—X3—CH2—, —(CH2)v—X3—CH2CH2— or —(CH2)w— unit in which each of the (CH2) groups is substituted by m radicals selected from the group consisting of halogen, methyl and (C1-C3)-alkoxy, or R7 and R8 together with the carbon atom to which they are bonded form the —O—N((C1-C3)-alkyl)-CHR10—CH2— or —O—N═CR10—CH2— unit in which each of the (CH2) groups is substituted by m radicals selected from the group consisting of halogen and methyl; R9 is hydrogen, (C1-C6)-alkyl, halo-(C1-C6)-alkyl, (C2-C6)-alkenyl, halo-(C2-C6)-alkenyl, (C2-C6)-alkynyl, halo-(C2-C6)-alkynyl, (C3-C7)-cycloalkyl, (C3-C7)-halocycloalkyl, (C3-C7)-cycloalkyl-(C1-C3)-alkyl, halo-(C3-C7)-cycloalkyl-(C1-C3)-alkyl, heteroaryl, heterocyclyl or phenyl, where the three latter radicals are each substituted by s radicals selected from the group consisting of halogen, nitro, cyano, (C1-C6)-alkyl, halo-(C1-C6) -alkyl, (C3-C6)-cycloalkyl, (C1-C6)-alkylthio, (C1-C6)-alkylsulfinyl, (C1-C6)-alkylsulfonyl, (C1-C6)-alkoxy, halo-(C1-C6)-alkoxy and (C1-C6)-alkoxy-(C1-C4)-alkyl; R10 is hydrogen, (C1-C3)-alkyl, or phenyl substituted by u radicals selected from the group Consisting of (C1-C3)-alkyl, halogen, cyano and nitro; R11 is hydrogen, (C1-C6)-alkyl, (C2-C6)-alkenyl, (C2-C6)-alkynyl, formyl, (C2-C6)-alkylcarbonyl, (C2-C6)-alkoxycarbonyl or (C1-C2)-alkylsulfonyl; X and Y are independently O, S, SO, SO2, C═O, C═S, NR10, CR7R8, C═NOR10 or C═NN(R11)2; X1 and X2 are each independently O, S or N((C1-C3)-alkyl); X3 is O or S; m is 0, 1 or 2; n is 2; r is 2, 3 or 4; s is 2, 3, 4 or 5; t is 1, 2, 3 or 4; u is 0, 1, 2 or 3; v is 2 or 3; and w is 2, 3, 4, 5 or 6. |
