发明名称 Purine inhibitors of human phosphatidylinositol 3-kinase delta
摘要 The instant invention provides compounds of formula I which are PI3K-delta inhibitors, and as such are useful for the treatment of PI3K-delta-mediated diseases such as inflamation, asthma, COPD and cancer.
申请公布号 AU2013347539(A1) 申请公布日期 2015.05.07
申请号 AU20130347539 申请日期 2013.11.15
申请人 MERCK SHARP & DOHME CORP. 发明人 ACHAB, ABDELGHANI ABE;ALTMAN, MICHAEL D.;DENG, YONGQI;KATTAR, SOLOMON;KATZ, JASON D.;METHOT, JOEY L.;ZHOU, HUA;MCGOWAN, MEREDETH;CHRISTOPHER, MATTHEW P.;GARCIA, YUDITH;ANTHONY, NEVILLE JOHN;FRADERA LLINAS, FRANCESC XAVIER;YANG, LIPING;MU, CHANGWEI;WANG, XIAONA;SHI, FENG;YE, BAIJUN;ZHANG, SIXING;ZHAO, XIAOLI;ZHANG, RONG;FONG, KIN CHIU;LENG, XIANSHENG
分类号 C07D473/34;A61K31/52;A61P11/00;A61P19/02;A61P35/00;A61P37/00 主分类号 C07D473/34
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