发明名称 |
INDOLE DERIVATIVES AS CRTH2 RECEPTOR ANTAGONISTS |
摘要 |
Compound of formula (I) are antagonists of the PGDreceptor, CRTH2, and as such are useful in the treatment and/or prevention of CRTH2-mediated diseases such as asthma. |
申请公布号 |
EA021076(B1) |
申请公布日期 |
2015.03.31 |
申请号 |
EA20110071081 |
申请日期 |
2010.02.19 |
申请人 |
MERCK SHARP & DOHME CORP.;MERCK CANADA INC. |
发明人 |
BERTHELETTE CARL;BOYD MICHAEL;COLUCCI JOHN;VILLENEUVE KARINE;METHOT JOEY |
分类号 |
C07D403/04;A61K31/405;A61K31/4192;A61K31/435;A61P11/06;C07D471/04 |
主分类号 |
C07D403/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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