发明名称 AN IMPROVED PROCESS FOR THE PURIFICATION OF BOCEPREVIR
摘要 The present invention relates to a process for the purification of Boceprevir, wherein hydroxyl Boceprevir is subjected to oxidation reaction in organic solvent after completion of the reaction, product is extracted into an aqueous bisulfate solution followed by pH adjustment to get pharmaceutically acceptable Boceprevir.
申请公布号 WO2015004685(A3) 申请公布日期 2015.03.12
申请号 WO2014IN00462 申请日期 2014.07.10
申请人 MYLAN LABORATORIES LTD;RAMA, SHANKAR;KAUSHIK, VIPIN KUMAR;RAVI, VIJAYA KRISHNA;RVN, VIKAS CHANDRADEV;MVSRK, CHAITANYA 发明人 RAMA, SHANKAR;KAUSHIK, VIPIN KUMAR;RAVI, VIJAYA KRISHNA;RVN, VIKAS CHANDRADEV;MVSRK, CHAITANYA
分类号 C07D209/52 主分类号 C07D209/52
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