发明名称 |
FUMARATE SALT OF (ALPHA S, BETA R)-6-BROMO-ALPHA-[2-(DIMETHYLAMINO)ETHYL]-2-METHOXY-ALPHA-1-NAPHTHALENYL-BETA-PHENYL-3-QUINOLINEETHANOL |
摘要 |
PROBLEM TO BE SOLVED: To provide a solid pharmaceutical composition for use in treatment or prevention of mycobacterial infection such as Mycobacterium tuberculosis.SOLUTION: The present invention relates to a solid pharmaceutical composition comprising fumarate salt of (alpha S, beta R)-6-bromo-alpha-[2-(dimethylamino)ethyl]-2-methoxy-alpha-1-naphthalenyl-beta-phenyl-3-quinolineethanol, and a humectant as polyethylene glycol sorbitan fatty acid ester. |
申请公布号 |
JP2015028049(A) |
申请公布日期 |
2015.02.12 |
申请号 |
JP20140191134 |
申请日期 |
2014.09.19 |
申请人 |
JANSSEN PHARMACEUTICA NV |
发明人 |
JEAN FRANCOIS ALEXANDRE HEGYI;WIM ALBERT ALEX AELTERMAN;YOLANDE LYDIA LANG;SIGRID CARL MARIA STOKBROEKX;CARINA LEYS;PETER JOZEF MARIA VAN REMOORTERE;ANNE FAURE |
分类号 |
A61K31/47;A61K9/20;A61K47/04;A61K47/12;A61K47/26;A61K47/34;A61K47/36;A61K47/38;A61P31/04;A61P31/06 |
主分类号 |
A61K31/47 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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