发明名称 DESFORMOTEROL AND PROCESS FOR ITS PREPARATION
摘要 The (R, R) -, (S, S) -, (R, S) -, ( DOLLAR I(R, S)) - isomers of 3 - amino- 4- hydroxy- alpha - [[[2- (4- methoxyphenyl)- 1-methylethyl]amino]methyl] -benzenemethanol (D) are disclosed, as well as an efficient method for their stereoselective synthesis. A method and composition are also disclosed utilizing desformoterol (D) as a bronchodilator, having high selectivity for beta 2 receptors.
申请公布号 WO9967198(A1) 申请公布日期 1999.12.29
申请号 WO1999US14082 申请日期 1999.06.22
申请人 SEPRACOR INC. 发明人 SENANAYAKE, CHRIS, HUGH
分类号 A61P11/08;A61K31/137;C07B61/00;C07C213/02;C07C213/04;C07C215/78;C07C217/60;C07C217/70 主分类号 A61P11/08
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