发明名称 |
NEW METHOD FOR PREPARING EZETIMIBE |
摘要 |
The present invention relates to a new method for preparing ezetimibe comprising a step of cyclizing the compound (4S)-phenyl-3-[(5S)-(4-fluorophenyl)-(2R)-[(1S)-(4-fluorophenylamino)-1-(4-nitrophenyl)methyl]-5-hydroxypentanoyl]oxazolidin-2-one or the derivatives thereof in which the hydroxyl group is protected. The invention also relates to new intermediates used in this method. |
申请公布号 |
HRP20141061(T1) |
申请公布日期 |
2015.01.02 |
申请号 |
HR2014P001061T |
申请日期 |
2014.11.03 |
申请人 |
MOEHS IBÉRICA, S.L. |
发明人 |
SÁNCHEZ CASALS, CARLES;DOBARRO RODRÍGUEZ, ALICIA;BOSCH CARTES, JUAN;GARCÍA DÍAZ, DAVINIA |
分类号 |
C07D205/08;C07D263/38 |
主分类号 |
C07D205/08 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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