发明名称 SOLUBILIZED CAPSULE FORMULATION OF 1,1-DIMETHYLETHYL [(1S)-1-{[(2S,4R)-4-(7-CHLORO-4METHOXYISOQUINOLIN-1-YLOXY)-2-({(1R,2S)-1-[(CYCLOPROPYLSULFONYL)CARBAMOYL]-2-ETHENYLCYCLOPROPYL}CARBAMOYL)PYRROLIDIN-1-YL]CARBONYL}-2,2-DIMETHYLPROPYL]CARBAMATE
摘要 <p>The present disclosure includes various embodiments directed to a solubilized capsule formulation of asunaprevir, 1,1-dimethylethyl[(1S)-1-{[(2S,4R)-4-(7-chloro-4methoxyisoquinolin-1-yloxy)-2-({(1R,2S)-1-[(cyclopropylsulfonyl)carbamoyl]-2-ethenylcyclopropyl}carbamoyl)pyrrolidin-1-yl]carbonyl}-2,2-dimethylpropyl]carbamate, and to methods including asunaprevir.</p>
申请公布号 SG11201406964Q(A) 申请公布日期 2014.11.27
申请号 SG11201406964Q 申请日期 2013.04.30
申请人 BRISTOL-MYERS SQUIBB HOLDINGS IRELAND 发明人 PERRONE, ROBERT KEVIN
分类号 A61K31/4709;A61K9/48;A61K31/4725;A61K38/06;A61P31/14 主分类号 A61K31/4709
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