发明名称 PROCESS FOR THE PREPARATION OF 2-CYANOPHENYLBORONIC ACID AND ESTERS THEREOF
摘要 The present invention relates to a process for the synthesis of 2-cyanophenylboronic acid and the esters and salts thereof of formula (II), which are intermediates of the synthesis of active pharmaceutical ingredients such as Perampanel or E2040. formula (II): (II).
申请公布号 EP2797931(A1) 申请公布日期 2014.11.05
申请号 EP20130745374 申请日期 2013.07.24
申请人 F.I.S.- FABBRICA ITALIANA SINTETICI S.P.A. 发明人 FONTANA, FRANCESCO;ROSSI, EMILIANO;DE FILIPPO, CHRISTIAN
分类号 C07F3/02;C07C253/30;C07D213/64;C07D295/155;C07F5/02;C07F5/04;C07F7/02 主分类号 C07F3/02
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