发明名称 ORGANIC COMPOUNDS
摘要 The present invention relates to optionally substituted 3-amino-4,5-dihydro-(1H or 2H)-pyrazolo[3,4-d]pyrimidin-6(7H)-ones and their 4-imino or 4-thioxo derivatives, e.g., 3-amino-4-(thioxo or imino)-4,5-dihydro-2H-pyrazolo[3,4-d]pyrimidin-6(7H)-ones, 3-amino-4-(thioxo or imino)-4,5-dihydro-2H-pyrazolo[3,4-d]pyrimidin-6(7H)-ones, 3-amino-4-(thioxo or imino)-4,5-dihydro-1H-pyrazolo[3,4-d]pyrimidin-6(7H)-ones, processes for their production, their use as pharmaceuticals and pharmaceutical compositions comprising them.
申请公布号 US2014315868(A1) 申请公布日期 2014.10.23
申请号 US201414252511 申请日期 2014.04.14
申请人 Intra-Cellular Therapies, Inc. 发明人 LI Peng;ZHAO Jun;ZHENG Hailin;WENNOGLE Lawrence
分类号 C07D487/04;A61K45/06;A61K31/519 主分类号 C07D487/04
代理机构 代理人
主权项 1. A 3-amino-(optionally 4-imino or 4-thioxo)-4,5-dihydro-(1H or 2H)-pyrazolo[3,4-d]pyrimidin-6-ones in free or salt form.
地址 New York NY US