发明名称 Compuestos derivados de aril dihidropiridinona y piperidinona como inhibidores de monoacilglicerol aciltransferasa (mgat2); composicion y combinacion farmaceutica; y uso en el tratamiento y prevencion de diabetes, hiperglucemia, retinopatia, sindrome metabolico, entre otras enfermedades.
摘要 The present invention provides compounds of Formula (I): or a stereoisomer, or a pharmaceutically acceptable salt thereof, wherein all of the variables are as defined herein. These compounds are monoacylglycerol acyltransferase type 2 (MGAT2) inhibitors which may be used as medicaments.
申请公布号 CL2014001437(A1) 申请公布日期 2014.10.03
申请号 CL20140001437 申请日期 2014.05.30
申请人 BRISTOL-MYERS SQUIBB COMPANY 发明人 TURDI, HUJI;HANGELAND, JON J.;LAWRENCE, R. MICHAEL;CHENG, DONG;AHMAD, SALEEM;MENG, WEI;BRIGANCE, ROBERT PAUL;DEVASTHALE, PRATIK;ZHAO, GUOHUA
分类号 C07D211/86;A61K31/4418;A61K31/4427;A61P3/00;C07D401/04;C07D401/14 主分类号 C07D211/86
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