发明名称 |
Compuestos derivados de aril dihidropiridinona y piperidinona como inhibidores de monoacilglicerol aciltransferasa (mgat2); composicion y combinacion farmaceutica; y uso en el tratamiento y prevencion de diabetes, hiperglucemia, retinopatia, sindrome metabolico, entre otras enfermedades. |
摘要 |
The present invention provides compounds of Formula (I):
or a stereoisomer, or a pharmaceutically acceptable salt thereof, wherein all of the variables are as defined herein. These compounds are monoacylglycerol acyltransferase type 2 (MGAT2) inhibitors which may be used as medicaments. |
申请公布号 |
CL2014001437(A1) |
申请公布日期 |
2014.10.03 |
申请号 |
CL20140001437 |
申请日期 |
2014.05.30 |
申请人 |
BRISTOL-MYERS SQUIBB COMPANY |
发明人 |
TURDI, HUJI;HANGELAND, JON J.;LAWRENCE, R. MICHAEL;CHENG, DONG;AHMAD, SALEEM;MENG, WEI;BRIGANCE, ROBERT PAUL;DEVASTHALE, PRATIK;ZHAO, GUOHUA |
分类号 |
C07D211/86;A61K31/4418;A61K31/4427;A61P3/00;C07D401/04;C07D401/14 |
主分类号 |
C07D211/86 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|