PROCESS AND INTERMEDIATES FOR THE PREPARATION OF PREGABALIN
摘要
The invention provides processes for the manufacture of a compound of formula (IA ). The invention further provides improved methods for the conversion of the compound of formula (I A ) into pregabalin.
申请公布号
CA2905411(A1)
申请公布日期
2014.10.02
申请号
CA20142905411
申请日期
2014.03.25
申请人
PFIZER IRELAND PHARMACEUTICALS
发明人
DEBARGE, SEBASTIEN;ERDMAN, DAVID THOMAS;O'NEILL, PADRAIG MARY;KUMAR, RAJESH;KARMILOWICZ, MICHAEL JOHN