发明名称 POLYMORPH FORM OF 4-{[4-({[4-(2,2,2-TRIFLUOROETHOXY)-1,2-BENZISOXAZOL-3-YL]OXY}METHYL)PIPERIDIN-1-YL]METHYL}-TETRAHYDRO-2H-PYRAN-4-CARBOXYLIC ACID
摘要 The present invention relates to novel crystal forms of 4-{[4-({[4-(2,2,2-trifluoroethoxy)-1,2-benzisoxazol-3-yl]oxy}methyl)piperidin-1-yl]methyl}-tetrahydro-2H-pyran-4-carboxylic acid. More particularly, the invention relates to polymorph forms (Polymorph Form I or Polymorph Form II), and to processes for the preparation of, compositions containing and to uses of, such polymorph forms.
申请公布号 EP2710002(A4) 申请公布日期 2014.10.01
申请号 EP20120786698 申请日期 2012.05.18
申请人 RAQUALIA PHARMA INC 发明人 NUMATA, TOYOHARU;NOGUCHI, HIROHIDE;WAIZUMI, NOBUAKI;KOJIMA, TAKASHI
分类号 C07D413/14;A61K31/454;A61P43/00 主分类号 C07D413/14
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