发明名称 |
POLYMORPH FORM OF 4-{[4-({[4-(2,2,2-TRIFLUOROETHOXY)-1,2-BENZISOXAZOL-3-YL]OXY}METHYL)PIPERIDIN-1-YL]METHYL}-TETRAHYDRO-2H-PYRAN-4-CARBOXYLIC ACID |
摘要 |
The present invention relates to novel crystal forms of 4-{[4-({[4-(2,2,2-trifluoroethoxy)-1,2-benzisoxazol-3-yl]oxy}methyl)piperidin-1-yl]methyl}-tetrahydro-2H-pyran-4-carboxylic acid. More particularly, the invention relates to polymorph forms (Polymorph Form I or Polymorph Form II), and to processes for the preparation of, compositions containing and to uses of, such polymorph forms. |
申请公布号 |
EP2710002(A4) |
申请公布日期 |
2014.10.01 |
申请号 |
EP20120786698 |
申请日期 |
2012.05.18 |
申请人 |
RAQUALIA PHARMA INC |
发明人 |
NUMATA, TOYOHARU;NOGUCHI, HIROHIDE;WAIZUMI, NOBUAKI;KOJIMA, TAKASHI |
分类号 |
C07D413/14;A61K31/454;A61P43/00 |
主分类号 |
C07D413/14 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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