发明名称 NOVEL PYRAZOLE DERIVATIVE
摘要 There has been a demand for a pharmaceutical composition which is used for a prophylactic and/or therapeutic agent for various diseases associated with PDE10 (for example, mental disorder, neurodegenerative disorder and the like). The present invention provides: a compound having a PDE10 inhibitory effect, in particular, a compound which is represented by formula (I) and is characterized by having a 4-heteroarylpyrazole-5-carboxylic acid amide structure, a pharmaceutically acceptable salt thereof, and a solvate of the compound or the salt; a pharmaceutical composition which is characterized by containing, as an active ingredient, the compound, a pharmaceutically acceptable salt of the compound, or a solvate of the compound or the salt; and a pharmaceutical use of the compound, a pharmaceutically acceptable salt of the compound, or a solvate of the compound or the salt.
申请公布号 WO2014133046(A1) 申请公布日期 2014.09.04
申请号 WO2014JP54773 申请日期 2014.02.26
申请人 MOCHIDA PHARMACEUTICAL CO., LTD. 发明人 OKANO AKIHIRO;SAITOH FUMIHIKO;MAKABE MUNEYOSHI;OGAWA KOUKI
分类号 C07D471/04;A61K31/444;A61K31/497;A61K31/506;A61K31/5377;A61P3/04;A61P25/00;A61P25/08;A61P25/14;A61P25/16;A61P25/18;A61P25/22;A61P25/24;A61P25/28;A61P25/32;A61P25/36;A61P43/00;C07D401/04;C07D417/04 主分类号 C07D471/04
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