发明名称 FUSED PHENYL AMIDO HETEROCYCLIC COMPOUNDS FOR THE PREVENTION AND TREATMENT OF GLUCOKINASE-MEDIATED DISEASES
摘要 The present invention relates to a compound of formula (VIa): or a pharmaceutically acceptable s alt or solvate thereof, wherein Ring A is pyrazinyl and L 1 , R 1 , R 1a , R 4 , L 2 , R 2 , R 3 , w and n are as defined herein. Such compounds are glucokinase agonists and useful in the treatment of diseases including diabetes and obesity.
申请公布号 PT2463283(E) 申请公布日期 2014.08.27
申请号 PT20120158318T 申请日期 2007.04.11
申请人 PFIZER PRODUCTS INC. 发明人 HAO BAI;SEIJI NUKUI;RU ZHOU;DILIP RAMAKANT BHUMRALKAR;FENG BI;FENGLI GUO;MINGYING HE;PAUL STUART HUMPHRIES;ANTHONY LAI LING;JIHONG LOU;SIMON BAILEY
分类号 C07D401/12;A61K31/41;A61K31/435;A61K31/495;C07D403/12;C07D405/12;C07D405/14;C07D409/12;C07D413/12;C07D413/14;C07D417/12;C07D417/14 主分类号 C07D401/12
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