发明名称 ESTROGEN RELATED RECEPTOR MODULATOR COMPOUND AND USE THEREOF
摘要 PROBLEM TO BE SOLVED: To provide a novel compound as an estrogen related receptor modulator used for treating metabolic disorders such as hyperlipemia, fatty liver, hyperglycemia, diabetes and obesity.SOLUTION: There is provided a compound of the formula I, a pharmaceutically acceptable salt thereof or a stereoisomer thereof. I, where A, B, D and E are independently CH or N, n is 0 to 2, a and b are o or 1, Ris H, a halogen, a hydroxyl group, a nitro group, a carboxyl group, a cyano group, an ester group, an amido group may be substituted and the like, Ris H, an alkyl group, an aryl group, a hetero ring and Ris H, a halogen, a hydroxyl group, a nitro group, a carboxyl group, a cyano group, an ester group, an amido group may be substituted.
申请公布号 JP2014141522(A) 申请公布日期 2014.08.07
申请号 JP20140080342 申请日期 2014.04.09
申请人 GUANGZHOU INSTITUTE OF BIOMEDICINE AND HEALTH CHINESE ACADEMY OF SCIENCES 发明人 DING KE;WONG CHIWAI;KANG ZHANFANG;ZHOU XI
分类号 C07D239/91;A61K31/517;A61K31/519;A61K31/5377;A61P1/16;A61P3/04;A61P3/06;A61P3/10;A61P9/10;A61P43/00;C07D471/04 主分类号 C07D239/91
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