发明名称 ROSUVASTATIN SALT, PROCESS FOR THE PREPARATION THEREOF AND PROCESS FOR THE PREPARATION OF PHARMACEUTICALLY ACCEPTABLE ROSUVASTATIN SALT
摘要 The invention relates to a salt of formula VIIwhere A isand Z is an amine of formula Zwhere R, Rand Rare independently selected from H, halogen, (C-C)alkyl, (C-C)alkoxy, CHF, CHFand CF, where halogen is independently selected from F, Cl, Br and I, and also to a process for preparing the same and to a process for preparing pharmaceutically acceptable rosuvastatin salt.
申请公布号 EA019995(B1) 申请公布日期 2014.07.30
申请号 EA20110090067 申请日期 2010.01.14
申请人 KRKA, TOVARNA ZDRAVIL, D.D., NOVO MESTO 发明人 BENKIC PRIMOZ;BEVK DAVID;LENARSIC ROMAN;ZUPANCIC SILVO;VAJS ANAMARIJA;JAKSE DAVID
分类号 C07D239/42 主分类号 C07D239/42
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