Process for the preparation of benzoimidazol-2-yl pyrimidine derivatives
摘要
The present invention is directed to processes for the preparation of benzoimidazol-2-yl pyrimidine derivatives useful as histamine H4 receptor modulators, and a crystalline hemi-tartrate of [5-(4,6-dimethyl-1H-benzoimidazol-2-yl)-4-methyl-pyrimidin-2-yl]-[3-(1-methyl-piperidin-4-yl)-propyl]-amine.
申请公布号
AU2009267159(B2)
申请公布日期
2014.05.15
申请号
AU20090267159
申请日期
2009.06.29
申请人
JANSSEN PHARMACEUTICA NV
发明人
MANI, NEELAKANDHA S.;CESCO-CANCIAN, SERGIO;PALMER, DAVID C.;LOCHNER, SUSANNE;XIAO, TONG;MAPES, CHRISTOPHER M.;GRIMM, JEFFREY S.;PIPPEL, DANIEL J.;BROGGINI, DIEGO