发明名称 |
SYNTHESIS AND NOVEL SALT FORMS OF (R)-3-((E)-2-(PYRROLIDIN-3-YL)VINYL)-5-(TETRAHYDROPYRAN-4-YLOXY)PYRIDINE |
摘要 |
The present invention relates to (R)-3-((E)-2-(pyrrolidin-3-yl)vinyl)-5-(tetrahydropyran-4-yloxy)pyridine, its salt forms, and to processes for the commercial-scale production of these compounds in sufficient purity and quality for use in pharmaceutical compositions. |
申请公布号 |
US2014107163(A1) |
申请公布日期 |
2014.04.17 |
申请号 |
US201314107175 |
申请日期 |
2013.12.16 |
申请人 |
TARGECEPT, INC. |
发明人 |
AKIREDDY SRINVASA RAO;BREINING SCOTT R.;CUTHBERTSON TIMOTHY J.;DULL GARY MAURICE;GATTO GREGORY J.;GENUS JOHN;HAMMOND PHILLIP S.;MITCHENER, JR. JOSEPH PIKE;MUNOZ JULIO A.;OTTEN PIETER ALBERT;YOHANNES DANIEL;FEDOROV NIKOLAI |
分类号 |
A61K31/4439 |
主分类号 |
A61K31/4439 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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