发明名称 Optionally substituted 3-amino-4-(thioxo or imino)-4,5-dihydro-2H-pyrazolo [3,4-d]pyrimidin-6(7H)-ones
摘要 The present invention relates to optionally substituted 3-amino-4,5-dihydro-(1H or 2H)-pyrazolo[3,4-d]pyrimidin-6(7H)-ones and their 4-imino or 4-thioxo derivatives, e.g., 3-amino-4-(thioxo or imino)-4,5-dihydro-2H-pyrazolo[3,4-d]pyrimidin-6(7H)-ones, 3-amino-4-(thioxo or imino)-4,5-dihydro-2H-pyrazolo[3,4-d]pyrimidin-6(7H)-ones, 3-amino-4-(thioxo or imino)-4,5-dihydro-1H-pyrazolo[3,4-d]pyrimidin-6(7H)-ones, processes for their production, their use as pharmaceuticals and pharmaceutical compositions comprising them.
申请公布号 US8697710(B2) 申请公布日期 2014.04.15
申请号 US200913132955 申请日期 2009.12.07
申请人 LI PENG;ZHAO JUN;ZENG HAILIN;WENNOGLE LAWRENCE;INTRA-CELLULAR THERAPIES, INC. 发明人 LI PENG;ZHAO JUN;ZENG HAILIN;WENNOGLE LAWRENCE
分类号 A01N43/90;A61K31/519;C07D487/00 主分类号 A01N43/90
代理机构 代理人
主权项
地址