发明名称 IMIDAZOTHIADIAZOLE DERIVATIVES AS PROTEASE ACTIVATED RECEPTOR 4 (PAR4) INHIBITORS FOR TREATING PLATELET AGGREGATION
摘要 <p>The present invention provides imidazothiadiazole compounds of Formula (I) wherein A, B, D, Rx, R1, R2, R3, X1, X2 and s are as defined herein, or a stereoisomer, tautomer, pharmaceutically acceptable salt or solvate form thereof, wherein all of the variables are as defined herein. These compounds are inhibitors of platelet aggregation and thus can be used as medicaments.</p>
申请公布号 WO2013163244(A8) 申请公布日期 2014.04.03
申请号 WO2013US37892 申请日期 2013.04.24
申请人 BRISTOL-MYERS SQUIBB COMPANY;UNIVERSITE DE MONTREAL 发明人 LAWRENCE, R. MICHAEL;MILLER, MICHAEL, M.;SEIFFERT, DIETMAR, ALFRED;POSY, SHOSHANA, L.;WONG, PANCRAS, C.;BANVILLE, JACQUES;RUEDIGER, EDWARD, H.;DEON, DANIEL, H.;MARTEL, ALAIN;TREMBLAY, FRANCOIS;GUY, JULIA;LAVALLEE, JEAN-FRANCOIS;GAGNON, MARC
分类号 C07D519/00;A61K31/433;A61K31/4439;A61P7/02;C07D513/04 主分类号 C07D519/00
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