发明名称 BICYCLIC HETEROCYCLE COMPOUNDS AND THEIR USES IN THERAPY
摘要 The invention relates to bicyclic heterocycle compounds of formula (I): or tautomeric or stereochemically isomeric forms, N-oxides, pharmaceutically acceptable salts or the solvates thereof; wherein R1, R2, R3, A, W, U and V are as defined herein; to pharmaceutical compositions comprising said compounds and to the use of said compounds in the treatment of diseases, e.g. cancer.
申请公布号 US2014045831(A1) 申请公布日期 2014.02.13
申请号 US201214112581 申请日期 2012.04.20
申请人 BUCK ILDIKO MARIA;CHESSARI GIANNI;HOWARD STEVEN;REES DAVID CHARLES;WOOLFORD ALISON JO-ANNE;ASTEX THERAPEUTICS LIMITED 发明人 BUCK ILDIKO MARIA;CHESSARI GIANNI;HOWARD STEVEN;REES DAVID CHARLES;WOOLFORD ALISON JO-ANNE
分类号 A61K31/5386;A61K31/437;A61K31/4985;A61K31/519;A61K31/5383;A61K45/06;C07D471/04;C07D498/04;C07D498/10 主分类号 A61K31/5386
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