发明名称 SULFONYL-DERIVATIVES AS NOVEL INHIBITORS OF HISTONE DEACETYLASE
摘要 This invention comprises the novel compounds of formula (I) wherein n, m, t, R1, R2, R3, R4, L, Q, X, Y, Z and have defined meanings, having histone deacetylase inhibiting enzymatic activity; their preparation, compositions containing them and their use as a medicine.
申请公布号 US2014038979(A1) 申请公布日期 2014.02.06
申请号 US201314053119 申请日期 2013.10.14
申请人 VAN EMELEN KRISTOF;ARTS JANINE;BACKX LEO-JACOBUS JOZEF;DE WINTER HANS LOUIS JOS;VAN BRANDT SVEN FRANCISCUS ANNA;VERDONCK MARC GUSTAAF CELINE;MEERPOEL LIEVEN;PILATTE ISABELLE NOELLE CONSTANCE;PONCELET VIRGINIE SOPHIE;DYATKIN ALEXEY BORISOVICH;VAN HEUSDEN JIMMY ARNOLD VIVIENE;JANSSEN PHARMACEUTICA NV 发明人 VAN EMELEN KRISTOF;ARTS JANINE;BACKX LEO-JACOBUS JOZEF;DE WINTER HANS LOUIS JOS;VAN BRANDT SVEN FRANCISCUS ANNA;VERDONCK MARC GUSTAAF CELINE;MEERPOEL LIEVEN;PILATTE ISABELLE NOELLE CONSTANCE;PONCELET VIRGINIE SOPHIE;DYATKIN ALEXEY BORISOVICH;VAN HEUSDEN JIMMY ARNOLD VIVIENE
分类号 C07D243/08;C07D295/26;A61K31/4545;A61K31/495;A61K31/496;A61K31/497;A61K31/501;A61K31/506;A61K31/52;A61K31/5377;A61K31/551;A61K45/06;A61P35/00;A61P43/00;C07D;C07D207/277;C07D207/28;C07D213/81;C07D213/82;C07D215/36;C07D233/34;C07D233/64;C07D233/84;C07D233/90;C07D237/24;C07D239/42;C07D239/48;C07D241/24;C07D241/26;C07D261/10;C07D295/22;C07D307/79;C07D333/34;C07D401/12;C07D403/04;C07D403/12;C07D405/12;C07D409/04;C07D409/12;C07D409/14;C07D413/12;C07D487/08;C07D513/04;G01N33/573 主分类号 C07D243/08
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