发明名称 |
NODULISPORIC ACID DERIVATIVE SPOT-ON FORMULATIONS FOR COMBATING PARASITES |
摘要 |
This invention provides for, inter alia, spot-on compositions for the treatment or prophylaxis of parasite infestations in mammals or birds which comprise: (1) at least one nodulisporic acid derivative; (2) an acceptable liquid carrier vehicle; and (3) optionally, a crystallization inhibitor. The invention also provides for a method of treating parasitic infestations or for the prophylaxis of parasite infestations in mammals or birds which comprise topically applying to said mammal or bird an effective amount of a composition according to the present invention. Further, this invention relates to an amidation process to prepare amide derivatives of nodulisporic acid and to intermediate formed in this process. |
申请公布号 |
CA2500822(C) |
申请公布日期 |
2013.12.24 |
申请号 |
CA20032500822 |
申请日期 |
2003.09.29 |
申请人 |
MERIAL LIMITED |
发明人 |
SOLL, MARK D.;BOECKH, ALBERT;DE BODE, RONUS;VAN EIJK, PETER JOHANNES SERVAAS SAVIO |
分类号 |
C07D491/052;A01N;A01N43/90;A61K;A61K9/00;A61K31/407;A61K31/475;C07D;C07D405/06;C07D491/14 |
主分类号 |
C07D491/052 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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