发明名称 |
Quinazolinones as inhibitors of human phosphatidylinositol 3-kinase delta |
摘要 |
The invention provides a class of substituted quinazolinone compounds and methods of treating diseases mediated by PI3Kdelta activity. The disclosed compounds are useful in treating diseases such as bone-resorption disorders; and cancer, especially hematopoietic cancers, lymphomas, multiple myelomas and leukemia. The compounds are also useful in disrupting or inhibiting cellular processes such as leukocyte function or accumulation, neutrophils function, lymphocyte proliferation, and endogenous immune responses. |
申请公布号 |
USRE44638(E1) |
申请公布日期 |
2013.12.10 |
申请号 |
US200513730256 |
申请日期 |
2005.05.12 |
申请人 |
FOWLER KERRY W.;HUANG DANWEN;KESICKI EDWARD A.;OOI HUA CHEE;OLIVER AMY;RUAN FUQIANG;TREIBERG JENNIFER;PURI KAMAL DEEP;ICOS CORPORATION |
发明人 |
FOWLER KERRY W.;HUANG DANWEN;KESICKI EDWARD A.;OOI HUA CHEE;OLIVER AMY;RUAN FUQIANG;TREIBERG JENNIFER;PURI KAMAL DEEP |
分类号 |
A61K31/517;A61K31/519;C07D239/91;C07D473/16;C07D473/34;C07D487/04 |
主分类号 |
A61K31/517 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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