发明名称 SUBSTITUTED INDOLYL ALKYL AMINO DERIVATIVES AS NOVEL INHIBITORS OF HISTONE DEACETYLASE
摘要 This invention comprises the novel compounds of formula (I) wherein R1, R2, R3, X and Y have defined meanings, having histone deacetylase inhibiting enzymatic activity; their preparation, compositions containing them and their use as a medicine.
申请公布号 US2013324568(A1) 申请公布日期 2013.12.05
申请号 US201313962523 申请日期 2013.08.08
申请人 VERDONCK MARC GUSTAAF CELINE;ANGIBAUD PARTICK RENE;ROUX BRUNO;PILATTE ISABELLE NOELLE CONSTANCE;TEN HOLTE PETER;ARTS JANINE;VAN EMELEN KRISTOF;JANSSEN PHARMACEUTICA N.V. 发明人 VERDONCK MARC GUSTAAF CELINE;ANGIBAUD PARTICK RENE;ROUX BRUNO;PILATTE ISABELLE NOELLE CONSTANCE;TEN HOLTE PETER;ARTS JANINE;VAN EMELEN KRISTOF
分类号 C07D401/14;A61K31/506;C07D405/14;C07D409/14;C07D491/056 主分类号 C07D401/14
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