发明名称 |
SUBSTITUTED INDOLYL ALKYL AMINO DERIVATIVES AS NOVEL INHIBITORS OF HISTONE DEACETYLASE |
摘要 |
This invention comprises the novel compounds of formula (I) wherein R1, R2, R3, X and Y have defined meanings, having histone deacetylase inhibiting enzymatic activity; their preparation, compositions containing them and their use as a medicine. |
申请公布号 |
US2013324568(A1) |
申请公布日期 |
2013.12.05 |
申请号 |
US201313962523 |
申请日期 |
2013.08.08 |
申请人 |
VERDONCK MARC GUSTAAF CELINE;ANGIBAUD PARTICK RENE;ROUX BRUNO;PILATTE ISABELLE NOELLE CONSTANCE;TEN HOLTE PETER;ARTS JANINE;VAN EMELEN KRISTOF;JANSSEN PHARMACEUTICA N.V. |
发明人 |
VERDONCK MARC GUSTAAF CELINE;ANGIBAUD PARTICK RENE;ROUX BRUNO;PILATTE ISABELLE NOELLE CONSTANCE;TEN HOLTE PETER;ARTS JANINE;VAN EMELEN KRISTOF |
分类号 |
C07D401/14;A61K31/506;C07D405/14;C07D409/14;C07D491/056 |
主分类号 |
C07D401/14 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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