发明名称 |
FUSED DIHYDROFURANS AS GPR119 MODULATORS FOR THE TREATMENT OF DIABETES, OBESITY AND RELATED DISORDERS |
摘要 |
<p>The present invention relates to compounds of general formula I, wherein the groups R1, LP, LQ, X1, X2, X3, A, n and m are as defined in the application. The compounds of formula I have valuable pharmacological properties, and in particular bind to the GPR119 receptor and modulate its activity.</p> |
申请公布号 |
EP2665719(A1) |
申请公布日期 |
2013.11.27 |
申请号 |
EP20120700413 |
申请日期 |
2012.01.20 |
申请人 |
BOEHRINGER INGELHEIM INTERNATIONAL GMBH |
发明人 |
HIMMELSBACH, FRANK;LANGKOPF, ELKE;NOSSE, BERND |
分类号 |
C07D407/14;A61K31/454;A61K31/4545;A61K31/497;A61K31/506;A61P3/10;A61P5/50;C07D413/14;C07D491/048 |
主分类号 |
C07D407/14 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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