发明名称 2,4-DIAMINO-6,7-DIHYDRO-5H-PYRROLO[2,3]PYRIMIDINE DERIVATIVES AS FAK/Pyk2 INHIBITORS
摘要 The invention relates to a novel class of 2,4-diamino-6,7-dihydro-5H-pyrrolo[2,3]pyrimidine derivatives as a FAK and/or Pyk2 inhibitor, to a process for their preparation, and to a composition thereof, as well as to use of the compounds for the inhibiting FAK and/or Pyk2 and method for the treatment of a FAK and/or Pyk2 mediated disorder or disease.
申请公布号 US2013281438(A1) 申请公布日期 2013.10.24
申请号 US201213978475 申请日期 2012.01.07
申请人 XIAO DENGMING;CHENG LIANG;LIU XIJIE;HU YUANDONG;XU XINHE;LIU ZHIHUA;ZHANG LIPENG;WU WEI;WANG SHULONG;SHEN YU;LI GEN;WANG YIN;ZHAO SHENG;LI CHONGLONG;TANG JIA;YU HONGHAO;CENTAURUS BIOPHARMA CO., LTD. 发明人 XIAO DENGMING;CHENG LIANG;LIU XIJIE;HU YUANDONG;XU XINHE;LIU ZHIHUA;ZHANG LIPENG;WU WEI;WANG SHULONG;SHEN YU;LI GEN;WANG YIN;ZHAO SHENG;LI CHONGLONG;TANG JIA;YU HONGHAO
分类号 C07D487/04 主分类号 C07D487/04
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