发明名称 |
2,4-DIAMINO-6,7-DIHYDRO-5H-PYRROLO[2,3]PYRIMIDINE DERIVATIVES AS FAK/Pyk2 INHIBITORS |
摘要 |
The invention relates to a novel class of 2,4-diamino-6,7-dihydro-5H-pyrrolo[2,3]pyrimidine derivatives as a FAK and/or Pyk2 inhibitor, to a process for their preparation, and to a composition thereof, as well as to use of the compounds for the inhibiting FAK and/or Pyk2 and method for the treatment of a FAK and/or Pyk2 mediated disorder or disease.
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申请公布号 |
US2013281438(A1) |
申请公布日期 |
2013.10.24 |
申请号 |
US201213978475 |
申请日期 |
2012.01.07 |
申请人 |
XIAO DENGMING;CHENG LIANG;LIU XIJIE;HU YUANDONG;XU XINHE;LIU ZHIHUA;ZHANG LIPENG;WU WEI;WANG SHULONG;SHEN YU;LI GEN;WANG YIN;ZHAO SHENG;LI CHONGLONG;TANG JIA;YU HONGHAO;CENTAURUS BIOPHARMA CO., LTD. |
发明人 |
XIAO DENGMING;CHENG LIANG;LIU XIJIE;HU YUANDONG;XU XINHE;LIU ZHIHUA;ZHANG LIPENG;WU WEI;WANG SHULONG;SHEN YU;LI GEN;WANG YIN;ZHAO SHENG;LI CHONGLONG;TANG JIA;YU HONGHAO |
分类号 |
C07D487/04 |
主分类号 |
C07D487/04 |
代理机构 |
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