发明名称 PROCESS FOR MAKING MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR
摘要 The invention provides a process for the preparation of a compound of Formula 1; comprising coupling a carboxylic acid of Formula 2; with an aniline of Formula 3; in the presence of a coupling agent. 0 0 No available figure
申请公布号 SG193156(A1) 申请公布日期 2013.09.30
申请号 SG20130057393 申请日期 2010.03.19
申请人 VERTEX PHARMACEUTICALS INCORPORATED 发明人 DEMATTEI, JOHN;LOOKER, ADAM, R.;NEUBERT-LANGILLE, BOBBIANNA;TRUDEAU, MARTIN;ROEPER, STEFANIE;RYAN, MICHAEL, P.;YAP, DAHRIKA, MILFRED LAO;KRUEGER, BRIAN, R.;GROOTENHUIS, PETER, D.J.;VAN GOOR, FREDERICK, F.;BOTFIELD, MARTYN, C.;ZLOKARNIK, GREGOR
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