发明名称 |
Radiolabelled Octreotate analogues as PET tracers |
摘要 |
Novel radiotracer(s) for Positron Emission Tomography (PET) imaging are described. Novel radiotracer(s) for Positron Emission Tomography (PET) imaging of neuorendocrine tumors are described. Specifically the present invention describes novel [18F]Fluoroethyltriazol-[Tyr3]Octreotate analogs; in particular those that target somatostatin receptors found on the cell surface of gastroenteropancreatic neuorendocrine tumors. The present invention also describes intermediate(s), precursor(s), pharmaceutical composition(s), methods of making, and methods of use of the novel radiotracer(s). |
申请公布号 |
AU2012223364(A1) |
申请公布日期 |
2013.09.19 |
申请号 |
AU20120223364 |
申请日期 |
2012.03.01 |
申请人 |
IMPERIAL COLLEGE;GE HEALTHCARE LIMITED |
发明人 |
LUTHRA, SAJINDER KAUR;LEYTON, JULIUS;ABOAGYE, ERIC OFORI;IDDON, LISA;INDREVOLL, BARD;GLASER, MATTHIAS EBERHARD;CUTHBERTSON, ALAN |
分类号 |
A61K51/08;A61K101/02;C07B59/00 |
主分类号 |
A61K51/08 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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